Monday 24 February 2014

Drug Induced Liver Disease (Hepatotoxicity)-Chapter 11-HISTOLOGICAL PATTERN IN DRUG-INDUCED LIVER DISEASE Part-4

Granulomatous hepatitis
        The most common causes of granulomas in the liver are infections, sarcoidosis, primary biliary cirrhosis and drugs.
        Granulomas are uncommon in hepatitis C but can occur in patients treated with interferon. Talc granulomas can occur in intravenous drug users and can be detected by viewing under polarised light. Other systemic granulomatous disease such as chronic metal toxicity (such as beryllium or copper) can also involve the liver. Finally, a study of granulomatous hepatitis cases over a 13-year period identified 11% as idiopathic. These cases can present with fever of unknown origin and generally respond favourably to steroids.
The granulomas can be present in the portal tracts or the parenchyma and lack necrosis. Unlike in primary biliary cirrhosis, the granulomas are not centred on the bile ducts. Granulomas also can occur with other patterns of liver injury such as acute hepatitis, cholestasis or steatosis.
         The term fibrin-ring granuloma has been used for small granulomas that consist of a ring of fibrin arranged around a central fat vacuole (fig 10). Epithelioid histiocytes are present around the ring of fibrin. In atypical cases, the fibrin is intermixed with the histiocytes and does not form a well-defined ring. More typical granulomas without the fibrin ring generally are present in other areas of the biopsy. Fibrin-ring granulomas have been described with allopurinol, BCG vaccination and intravesical therapy for carcinoma. These granulomas were first described in the rickettsial disease Q fever (Coxiella burnetti) but also occur in boutonneuse fever (Rickettsia conorii), leishmaniasis, toxoplasmosis, cytomegalovirus infection and Hodgkin lymphoma.

Steatosis and steatohepatitis
Macrovesicular steatosis
        Macrovesicular steatosis includes large and small droplet fat. The term “large droplet fat” is used when at least half the hepatocyte cytoplasm is occupied by a single lipid vacuole, while multiple lipid vacuoles are seen in small droplet fat. The latter often is confused with true microvesicular steatosis which, unlike small droplet fat, affects the liver in a diffuse fashion. Macrovesicular steatosis can be seen in association with steroids, nitrofurantoin, gold, methotrexate, NSAIDs such as ibuprofen, indomethacin and sulindac, and antihypertensives such as metoprolol, chlorinated hydrocarbons such as carbon tetrachloride and chloroform, or chemotherapeutic agents such as 5-fluorouracil, cisplatin and tamoxifen.
Microvesicular steatosis
        Exclusive or predominant microvesicular steatosis diffusely affecting the liver is a result of mitochondrial injury and often occurs as an adverse effect of drugs/toxins such as cocaine, tetracycline, valproic acid and zidovudine (fig 11). Acute exposure to alcohol (alcohol foamy liver degeneration) and paediatric Reye syndrome also show diffuse microvesicular steatosis. Other non-drug related aetiologies include acute fatty liver of pregnancy and genetic diseases such as carnitine deficiency.

Steatohepatitis
By definition, steatohepatitis is characterised by steatosis, lobular inflammation and hepatocellular injury in the form of hepatocellular ballooning (with or without acidophil bodies or Mallory hyaline) or pericellular fibrosis. A few drugs (notably amiodarone and irinotecan) play a direct aetiological role in steatohepatitis. Most other drugs exacerbate or precipitate steatohepatitis in the presence of other risk factors such as obesity and diabetes.
Amiodarone
Amiodarone, a potent antiarrhythmic agent, causes elevated liver enzymes in up to 30% of patients and steatohepatitis in 1–2%  of patients. Amiodarone steatohepatitis is characterised by prominent Mallory hyaline (occasionally in zone 1) and neutrophilic satellitosis, while steatosis is less conspicuous (fig 12). It is also associated with a different type of lipid accumulation called “phospholipidosis” characterised by accumulation of drug in the lysosomes.  This leads to “foamy” appearance of hepatocytes and Kupffer cells. The foamy areas show lamellar lysosomal inclusion bodies on electron microscopy (fig 13).
Chemotherapy-induced steatohepatitis
Steatosis and steatohepatitis have been reported with chemotherapeutic agents. The latter especially is associated with irinotecan, a drug often used preoperatively in colorectal cancer with hepatic metastases. This has been referred to as chemotherapy-associated steatohepatitis in the oncology literature. Other chemotherapeutic agents such as oxaliplatin have been variably implicated.
Vascular abnormalities
Several vascular patterns of injury are recognised, each with distinctive morphological features and drug associations.
Sinusoidal obstruction syndrome
Sinusoidal obstruction syndrome (SOS; veno-occlusive disease) is due to endothelial cell injury to small hepatic venules that manifests histologically as endothelial swelling and thrombosis (fig 14). The resultant venous outflow obstruction leads to sinusoidal dilatation, congestion, hepatocellular necrosis, and can result in centrilobular fibrosis. Cytotoxic/chemotherapeutic drugs such as oxaliplatin (used in colorectal cancer) can cause injury to sinusoidal endothelial cells and hepatic stellate cells.
Peliosis hepatis
        Peliosis is characterised by blood-filled cavities without an endothelial lining in the hepatic parenchyma (fig 15). This phenomenon most commonly is associated with androgens or contraceptive steroids. Thiopurine-derived chemotherapeutic drugs also have been implicated. Peliosis also occurred with the intravenous contrast agent thorium dioxide (Thorotrast), which has been discontinued due to the high risk of angiosarcoma. Sinusoidal dilatation may accompany peliosis or may occur independently, particularly with androgenic or oestrogenic steroid use.

Hepatic vein thrombosis
Hepatic vein thrombosis is a rare complication of some drugs, including oral contraceptives and dacarbazine, and presents clinically as Budd-Chiari syndrome.

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